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Synthesis of unnatural amino acids and other blocks

Icotrokinra

Name
Icotrokinra
Molecular structural formula
Purity
≥98%
CAS Number
2763602-16-8
Formula
C90H120N20O22S2
MW
1898.17
Target
Interleukin Related STAT
Sequence
Ac-Pen-Asn-Thr-Trp(7-Me)-Lys(Ac)-Pen-Phe(4-amino ethoxy)-2Nal-ThpGly-Glu-Asn-3Pal-Sar-NH2 (Pen1&Pen6 bridge)
Sequence Shortening
Ac-Pen-NT-Trp(7-Me)-Lys(Ac)-Pen-Phe(4-amino ethoxy)-2Nal-ThpGly-EN-3Pal-Sar-NH2 (Pen1&Pen6 bridge)
InChIKey
IVFNYXYPMJQSGF-QMRCQSNESA-N
Solubility in DMSO
100 mg/mL
References
[1]. Fourie AM, et al., JNJ-77242113, a highly potent, selective peptide targeting the IL-23 receptor, provides robust IL-23 pathway inhibition upon oral dosing in rats and humans. Sci Rep. 2024 Jul 30;14(1):17515.
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Product details
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Icotrokinra, an oral IL-23 receptor antagonist, has been shown to effectively block IL-23-mediated STAT3 phosphorylation and IFN-γ production in NK cells, showing significant anti-inflammatory effects. This drug mainly acts on the IL-23 receptor in the process of pathogenic T cell activation in plaque psoriasis, so it has potential application value in the research fields of psoriasis, psoriatic arthritis and inflammatory bowel disease.