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Cortistatin 17, human

Name
Cortistatin 17, human
Molecular structural formula
Purity
≥95%
Price

1mg: $42.00

5mg: $129.50

10mg: $213.50

CAS Number
189450-19-9
Formula
C96H139N27O24S3
MW
2151.54
Target
others
Sequence
Asp-Arg-Met-Pro-Cys-Arg-Asn-Phe-Phe-Trp-Lys-Thr-Phe-Ser-Ser-Cys-Lys (Disulfide bridge Cys5-Cys16)
Sequence Shortening
DRMPCRNFFWKTFSSCK(Disulfide bridge Cys5-Cys16)
InChIKey
GRHDFHUELYLPDB-XOJLFHOJSA-N
References
[1].Convenient fluorometric assay for matrix metalloproteinase activity and its application in biological media.B.Beekman et al., FEBS Lett., 390, 221 (1996) [2].Identification and characterization of a novel human cortistatin-like peptide.S.Fukusumi et al., Biochem. Biophys. Res. Commun., 232, 157 (1997)
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Product details
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Cortistatin-17 shows structural similarities to somatostatin. The peptide binds to all somatostatin receptor subtypes (SSTR) in a similar way as the rat cortistatin. Its inhibitory effects on forskolin-stimulated cAMP production in chinese hamster ovary cells expressing SSTR2-5 are dose dependent but slightly less efficient than that of somatostatin-14. Like the rat cortistatin it has an effect on sleep and wakefulness pattern in rat. It decreases the light slow wave sleep (SWS1) and increases the deep slow wave sleep (SWS2) in a dose dependent manner. Administration of the peptide causes a temporary flattening of cortical and hippocampal electroencephalograms.